Tamoxifen citrate，Estrogen receptor拮抗剂and partial激动剂(ab120656)
Key features and details
- Estrogen receptor antagonist and partial agonist
- CAS Number: 54965-24-1
- Purity: > 99%
- Soluble in DMSO to 100 mM and in ethanol to 5 mM
- Form / State: Solid
- Source: Synthetic
概述
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产品名称
Tamoxifen citrate，Estrogen receptor拮抗剂and partial激动剂 -
描述
Estrogen receptor拮抗剂and partial激动剂 -
生物学描述
Competitive estrogen receptor antagonist and partial agonist. Inhibits estrogen dependent gene transcription and tumor growth. Additionally decreases cardiac infarction and inhibits Kir2.1, Kir2.2 and Kir2.3 potassium channels (IC50 values are 0.93, 0.87 and 0.31 µM, respectively).
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纯度
> 99% -
CAS编号
54965-24-1 -
化学结构
性能
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化学名称
(Z)-2-[4-(1,2-Diphenyl-1-butenyl)phenoxy]-N,N-dimethylethanamine citrate -
分子量
563.65 -
分子式
C26H29NO.C6H8O7 -
存放说明
Store at +4°C. The product can be stored for up to 12 months. -
溶解度概述
Soluble in DMSO to 100 mM and in ethanol to 5 mM -
处理
Wherever possible, you should prepare and use solutions on the same day. However, if you need to make up stock solutions in advance, we recommend that you store the solution as aliquots in tightly sealed vials at -20°C. Generally, these will be useable for up to one month. Before use, and prior to opening the vial we recommend that you allow your product to equilibrate to room temperature for at least 1 hour.
Toxic, refer to SDS for further information
Need more advice on solubility, usage and handling? Please visit our frequently asked questions (FAQ) page for more details.
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来源
Synthetic
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研究领域
图片
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Chemical Structure - Tamoxifen citrate, Estrogen receptor antagonist and partial agonist (ab120656)2D chemical structure image of ab120656, Tamoxifen citrate, Estrogen receptor antagonist and partial agonist
实验方案
To our knowledge, customised protocols are not required for this product. Please try the standard protocols listed below and let us know how you get on.
文献 (0)
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