CGP 7930，Positive allosteric modulator of GABAB receptors (ab120492)
Key features and details
- Positive GABAB receptor allosteric modulator
- CAS Number: 57717-80-3
- Soluble in DMSO to 100 mM and in ethanol to 100 mM
- Form / State: Solid
- Source: Synthetic
概述
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产品名称
CGP 7930，Positive allosteric modulator of GABAB receptors -
描述
Positive GABAB receptor allosteric modulator -
生物学描述
Positive GABAB receptor allosteric modulator (EC50 values are 5.37 and 4.60 μM, respectively). Increases receptor agonist affinity and signal transduction efficacy. Also shown to potentiate receptor response to baclofen (ab120325).
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CAS编号
57717-80-3 -
化学结构
性能
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化学名称
3,5-Bis(1,1-dimethylethyl)-4-hydroxy-β,β-dimethylbenzenepropanol -
分子量
292.46 -
分子式
C19H32O2 -
PubChem识别号
5024764 -
存放说明
Store at Room Temperature. Store under desiccating conditions. The product can be stored for up to 12 months. -
溶解度概述
Soluble in DMSO to 100 mM and in ethanol to 100 mM -
处理
Wherever possible, you should prepare and use solutions on the same day. However, if you need to make up stock solutions in advance, we recommend that you store the solution as aliquots in tightly sealed vials at -20°C. Generally, these will be useable for up to one month. Before use, and prior to opening the vial we recommend that you allow your product to equilibrate to room temperature for at least 1 hour.
Need more advice on solubility, usage and handling? Please visit our frequently asked questions (FAQ) page for more details.
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SMILES
CC(C)(C)c1cc(cc(c1O)C(C)(C)C)CC(C)(C)CO -
来源
Synthetic
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研究领域
相关产品
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图片
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Chemical Structure - CGP 7930, Positive allosteric modulator of GABAB receptors (ab120492)2D chemical structure image of ab120492, CGP 7930, Positive allosteric modulator of GABAB receptors
实验方案
To our knowledge, customised protocols are not required for this product. Please try the standard protocols listed below and let us know how you get on.
文献 (0)
ab120492 尚未被引用在任何文献中。