BRL 44408 maleate，alpha2A adrenoceptor拮抗剂(ab120806)
Key features and details
- Selective α2A adrenoceptor antagonist
- CAS Number: 681806-46-2
- Purity: > 99%
- Soluble in water to 100 mM
- Form / State: Solid
- Source: Synthetic
概述
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产品名称
BRL 44408 maleate，alpha2A adrenoceptor拮抗剂 -
描述
Selective α2A adrenoceptor拮抗剂 -
生物学描述
Selective α2A adrenoceptor antagonist (Ki values are 5.68 and 651 nM for α2A and α2B, respectively). Centrally active following subcutaneous administration. Demonstrates antidepressant and analgesic activity.
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纯度
> 99% -
CAS编号
681806-46-2 -
化学结构
性能
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化学名称
2-[(4,5-Dihydro-1H-imidazol-2-yl)methyl]-2,3-dihydro-1-methyl-1H-isoindole maleate -
分子量
331.37 -
分子式
C13H17N3.C4H4O4 -
存放说明
Store at -20°C. Store under desiccating conditions. The product can be stored for up to 12 months. -
溶解度概述
Soluble in water to 100 mM -
处理
Wherever possible, you should prepare and use solutions on the same day. However, if you need to make up stock solutions in advance, we recommend that you store the solution as aliquots in tightly sealed vials at -20°C. Generally, these will be useable for up to one month. Before use, and prior to opening the vial we recommend that you allow your product to equilibrate to room temperature for at least 1 hour.
Need more advice on solubility, usage and handling? Please visit our frequently asked questions (FAQ) page for more details.
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来源
Synthetic
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研究领域
图片
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Chemical Structure - BRL 44408 maleate, alpha2A adrenoceptor antagonist (ab120806)2D chemical structure image of ab120806, BRL 44408 maleate, alpha2A adrenoceptor antagonist
实验方案
To our knowledge, customised protocols are not required for this product. Please try the standard protocols listed below and let us know how you get on.
文献 (1)
ab120806 被引用在 1 文献中.
- Li Q et al. Sympathetic Denervation Ameliorates Renal Fibrosis via Inhibition of Cellular Senescence. Front Immunol 12:823935 (2021). PubMed: 35140713