概述

  • 产品名称
    Varenicline tartrate
  • 描述
    Orally active partial agonist at α4β2 nicotinic receptors
  • 生物学描述
    High affinity, subtype-selective partial agonist at α4β2 nicotinic receptors. (Ki values are 0.06 (α4β2), 240 (α3β4), 322 (α7) and 3540 nM (α1βγδ)). Full agonist at α7 receptors. Orally active.
  • 纯度
    > 99%

性能

  • 化学名称
    7,8,9,10-Tetrahydro-6,10-methano-6H-pyrazino[2,3-h][3]benzazepine tartrate
  • 分子量
    361.37
  • 化学结构
    Chemical Structure
  • 分子式
    C13H13N3.C4H6O6
  • CAS编号
    375815-87-5
  • 存放说明
    Store at Room Temperature. Store under desiccating conditions. The product can be stored for up to 12 months.
  • 溶解度概述
    Soluble in water to 100 mM
  • 处理

    Wherever possible, you should prepare and use solutions on the same day. However, if you need to make up stock solutions in advance, we recommend that you store the solution as aliquots in tightly sealed vials at -20°C. Generally, these will be useable for up to one month. Before use, and prior to opening the vial we recommend that you allow your product to equilibrate to room temperature for at least 1 hour.

    Need more advice on solubility, usage and handling? Please visit our frequently asked questions (FAQ) page for more details.

  • 来源

    Synthetic

  • 研究领域

    Varenicline tartrate (ab120539)参考文献

    This product has been referenced in:

    See all 4 Publications for this product

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