GS 39783,GABAB positive allosteric modulator (ab120320)
Key features and details
- Novel, GABAB positive allosteric modulator
- CAS Number: 39069-52-8
- Purity: > 99%
- Soluble in DMSO to 25 mM
- Form / State: Solid
- Source: Synthetic
概述
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产品名称
GS 39783,GABAB positive allosteric modulator -
描述
Novel,GABAB positive allosteric modulator -
生物学描述
Novel, GABAB positive allosteric modulator (EC50 = 3 μM for [35S]GTPγS binding). Shows anxiolytic and antiaddictive effects in vivo. Blood-brain barrier permeable. Orally active.
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纯度
> 99% -
CAS编号
39069-52-8 -
化学结构
性能
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化学名称
N4,N6-Dicyclopentyl-2-(methylthio)-5-nitro-4,6-pyrimidinediamine -
分子量
337.44 -
分子式
C15H23N5O2S -
PubChem识别号
6604928 -
存放说明
Store at -20°C. Store In the Dark. Store under desiccating conditions. This product is air and light sensitive and impurities can occur as a result of air oxidation or due to metabolism by microbes. -
溶解度概述
Soluble in DMSO to 25 mM -
处理
Wherever possible, you should prepare and use solutions on the same day. However, if you need to make up stock solutions in advance, we recommend that you store the solution as aliquots in tightly sealed vials at -20°C. Generally, these will be useable for up to one month. Before use, and prior to opening the vial we recommend that you allow your product to equilibrate to room temperature for at least 1 hour.
Refer to SDS for further information
Need more advice on solubility, usage and handling? Please visit our frequently asked questions (FAQ) page for more details.
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SMILES
CSC1=NC(=C(C(=N1)NC2CCCC2)[N+](=O)[O-])NC3CCCC3 -
来源
Synthetic
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研究领域
实验方案
To our knowledge, customised protocols are not required for this product. Please try the standard protocols listed below and let us know how you get on.
文献 (0)
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