Selective δ opioid receptor agonist (Ki values are 1.5, >1000 and >1000 nM for opioid receptor subtypes δ, μ and κ, respectively). Antinociceptive activity. Centrally active following intravenous administration.
Store at -20°C. Store under desiccating conditions. The product can be stored for up to 12 months.
Soluble in water to 0.5 mg/ml
Wherever possible, you should prepare and use solutions on the same day. However, if you need to make up stock solutions in advance, we recommend that you store the solution as aliquots in tightly sealed vials at -20°C. Generally, these will be useable for up to one week. Before use, and prior to opening the vial we recommend that you allow your product to equilibrate to room temperature for at least 1 hour.
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Toll L et al. Standard binding and functional assays related to medications development division testing for potential cocaine and opiate narcotic treatment medications. NIDA Res Monogr178:440-66 (1998).
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