SB 271046 hydrochloride,5-HT6拮抗剂(ab120589)
Key features and details
- Potent, selective 5-HT6 antagonist
- CAS Number: 209481-24-3
- Purity: > 99%
- Soluble in DMSO to 100 mM and in ethanol to 5 mM (with heating)
- Form / State: Solid
- Source: Synthetic
概述
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产品名称
SB 271046 hydrochloride,5-HT6拮抗剂 -
描述
Potent,selective 5-HT6拮抗剂 -
生物学描述
Potent and selective 5-HT6 receptor antagonist (Ki = 1-2 nM). Displays >200-fold selectivity for 5-HT6 receptors (vs. other receptor binding sites and ion channels). Poor penetration of the blood-brain barrier. Nootropic effects in vivo.
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纯度
> 99% -
CAS编号
209481-24-3 -
化学结构
性能
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化学名称
5-Chloro-N-[4-methoxy-3-(1-piperazinyl)phenyl]-3-methylbenzo[b]thiophen-2-sulfonamide hydrochloride -
分子量
488.45 -
分子式
C20H22CIN3O3S2.HCl -
存放说明
Store at +4°C. Store under desiccating conditions. The product can be stored for up to 12 months. -
溶解度概述
Soluble in DMSO to 100 mM and in ethanol to 5 mM (with heating) -
处理
Wherever possible, you should prepare and use solutions on the same day. However, if you need to make up stock solutions in advance, we recommend that you store the solution as aliquots in tightly sealed vials at -20°C. Generally, these will be useable for up to one month. Before use, and prior to opening the vial we recommend that you allow your product to equilibrate to room temperature for at least 1 hour.
Need more advice on solubility, usage and handling? Please visit our frequently asked questions (FAQ) page for more details.
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来源
Synthetic
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研究领域
实验方案
To our knowledge, customised protocols are not required for this product. Please try the standard protocols listed below and let us know how you get on.
文献 (0)
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