BMY 7378 dihydrochloride,5-HT1A partial激动剂. alpha adrenoceptor拮抗剂. (ab120520)
Key features and details
- 5-HT1A partial agonist. α adrenoceptor antagonist.
- CAS Number: 21102-95-4
- Purity: > 99%
- Soluble in water to 100 mM
- Form / State: Solid
- Source: Synthetic
概述
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产品名称
BMY 7378 dihydrochloride,5-HT1A partial激动剂. alpha adrenoceptor拮抗剂. -
描述
5-HT1A partial激动剂. α adrenoceptor拮抗剂. -
生物学描述
5-HT1A partial agonist (IC50 = 0.8 nM). Potent and selective α1D adrenoceptor antagonist (Ki values are 2, 600 and 800 nM at α1D, α1B and α1A receptors, respectively). Shows antihypertensive activity.
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纯度
> 99% -
CAS编号
21102-95-4 -
化学结构
性能
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化学名称
8-[2-[4-(2-Methoxyphenyl)-1-piperazinyl]ethyl]-8-azaspirol[4,5]decane-7,9-dione dihydrochloride -
分子量
458.43 -
分子式
C22H31N3O3.2HCl -
存放说明
Store at Room Temperature. The product can be stored for up to 12 months. -
溶解度概述
Soluble in water to 100 mM -
处理
Wherever possible, you should prepare and use solutions on the same day. However, if you need to make up stock solutions in advance, we recommend that you store the solution as aliquots in tightly sealed vials at -20°C. Generally, these will be useable for up to one month. Before use, and prior to opening the vial we recommend that you allow your product to equilibrate to room temperature for at least 1 hour.
Need more advice on solubility, usage and handling? Please visit our frequently asked questions (FAQ) page for more details.
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来源
Synthetic
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研究领域
图片
实验方案
To our knowledge, customised protocols are not required for this product. Please try the standard protocols listed below and let us know how you get on.
文献 (0)
ab120520 尚未被引用在任何文献中。