2-Chloro-N6-cyclopentyladenosine (CCPA) (ab120434)

概述

  • 产品名称2-Chloro-N6-cyclopentyladenosine (CCPA)
  • 描述
    Highly potent, selective A1 agonist
  • 别名
    • CCPA
  • 生物学描述Highly potent and selective A1 receptor agonist (Ki values are 0.8, 2300 and 42 nM for human A1, A2A and A3 receptors, respectively). Shows >2000-fold selectivity over A2A. Centrally active following systemic administration and anticonvulsive in vivo.
  • 纯度> 98%

性能

    2-Chloro-N6-cyclopentyladenosine (CCPA) (ab120434)参考文献

    This product has been referenced in:
    • Monopoli A  et al. Pharmacology of the highly selective A1 adenosine receptor agonist 2-chloro-N6-cyclopentyladenosine. Arzneimittelforschung 44:1305-12 (1994). Read more (PubMed: 7848348) »
    • Lohse MJ  et al. 2-Chloro-N6-cyclopentyladenosine: a highly selective agonist at A1 adenosine receptors. Naunyn Schmiedebergs Arch Pharmacol 337:687-9 (1988). Read more (PubMed: 3216901) »
    • Luszczki JJ  et al. 2-Chloro-N6-cyclopentyladenosine enhances the anticonvulsant action of carbamazepine in the mouse maximal electroshock-induced seizure model. Pharmacol Rep 57:787-94 (0). Read more (PubMed: 16382198) »

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    The datasheet for this product states that it is soluble in water to 5 mM, this indicates that it should also be soluble in PBS or saline.



    Depending on the assay, I would also advi...

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    Thank you for your email last week and for your patience while I have been in touch with the lab about your enquiry.

    The compound contains 0.5 moles of water per mole of compound. This equates to 2.38% water by weight.

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